Eptapirone
Eptapirone is a potent and highly selective 5-HT1A receptor full agonist of the azapirone chemical class. It is an anxiolytic drug that was first synthesized by Bristol-Myers Squibb in 1986. Eptapirone is structurally related to other azapirones like buspirone and ipsapirone.
Pharmacology
Eptapirone acts as a full agonist at the 5-HT1A receptor, meaning it can produce the maximum response possible from this receptor. This is in contrast to partial agonists, which can only produce a partial response regardless of the drug dosage. The 5-HT1A receptor is a subtype of the 5-HT receptor that binds the neurotransmitter serotonin, and is involved in a variety of functions including mood, anxiety, and cognition.
Clinical Use
Eptapirone has been studied for its potential use in the treatment of anxiety disorders, depression, and other conditions. However, as of 2021, it is not currently approved for medical use in any country.
Chemistry
Eptapirone belongs to the azapirone class of compounds, which are characterized by their pyrimidinylpiperazine and furanopyridine moieties. Other azapirones include buspirone, gepirone, and ipsapirone, all of which also act as 5-HT1A receptor agonists.
See Also
References
Transform your life with W8MD's budget GLP-1 injections from $125.
W8MD offers a medical weight loss program to lose weight in Philadelphia. Our physician-supervised medical weight loss provides:
- Most insurances accepted or discounted self-pay rates. We will obtain insurance prior authorizations if needed.
- Generic GLP1 weight loss injections from $125 for the starting dose.
- Also offer prescription weight loss medications including Phentermine, Qsymia, Diethylpropion, Contrave etc.
NYC weight loss doctor appointments
Start your NYC weight loss journey today at our NYC medical weight loss and Philadelphia medical weight loss clinics.
- Call 718-946-5500 to lose weight in NYC or for medical weight loss in Philadelphia 215-676-2334.
- Tags:NYC medical weight loss, Philadelphia lose weight Zepbound NYC, Budget GLP1 weight loss injections, Wegovy Philadelphia, Wegovy NYC, Philadelphia medical weight loss, Brookly weight loss and Wegovy NYC
|
WikiMD's Wellness Encyclopedia |
| Let Food Be Thy Medicine Medicine Thy Food - Hippocrates |
Medical Disclaimer: WikiMD is not a substitute for professional medical advice. The information on WikiMD is provided as an information resource only, may be incorrect, outdated or misleading, and is not to be used or relied on for any diagnostic or treatment purposes. Please consult your health care provider before making any healthcare decisions or for guidance about a specific medical condition. WikiMD expressly disclaims responsibility, and shall have no liability, for any damages, loss, injury, or liability whatsoever suffered as a result of your reliance on the information contained in this site. By visiting this site you agree to the foregoing terms and conditions, which may from time to time be changed or supplemented by WikiMD. If you do not agree to the foregoing terms and conditions, you should not enter or use this site. See full disclaimer.
Credits:Most images are courtesy of Wikimedia commons, and templates, categories Wikipedia, licensed under CC BY SA or similar.
Contributors: Prab R. Tumpati, MD
