Ro4938581
Ro4938581 is a pharmacological compound that acts as a positive allosteric modulator at the GABAA receptor. It is a derivative of the benzodiazepine class of drugs, with a unique chemical structure that distinguishes it from other benzodiazepines.
Chemistry
Ro4938581 is a benzodiazepine derivative, meaning it is structurally related to drugs such as diazepam and alprazolam. However, unlike these drugs, Ro4938581 has a unique chemical structure that includes a pyrazoloquinolinone core, which is not found in other benzodiazepines. This unique structure is thought to contribute to its distinct pharmacological properties.
Pharmacology
Ro4938581 acts as a positive allosteric modulator at the GABAA receptor, a type of ionotropic receptor that is widely distributed throughout the central nervous system. By enhancing the activity of this receptor, Ro4938581 can increase the inhibitory effects of the neurotransmitter GABA, which can lead to sedative, anxiolytic, and anticonvulsant effects.
Clinical Use
While Ro4938581 has been studied in preclinical trials, it has not yet been approved for use in humans. However, its unique pharmacological properties make it a promising candidate for the treatment of conditions such as anxiety disorders, insomnia, and epilepsy.
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Contributors: Prab R. Tumpati, MD
